Publications
2022 Heading link
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25th January, 2022
XP-524 is a dual-BET/EP300 inhibitor that represses oncogenic KRAS and potentiates immune checkpoint inhibition in pancreatic cancer
Authors:
Daniel R. Principe, Rui Xiong, Yangfeng Li, Thao N. D. Pham, Suneel D. Kamath, Oleksii Dubrovskyi, Kiira Ratia, Fei Huang, Jiong Zhao, Zhengnan Shen, Dinesh Thummuri, Zhou Daohong, Patrick W. Underwood, Jose Trevino, Hidayatullah G. Munshi, Gregory R. J. Thatcher, and Ajay RanaJournal:
PNAS -
24th January, 2022
Structure–Activity Relationships and Transcriptomic Analysis of Hypoxia-Inducible Factor Prolyl Hydroxylase Inhibitors
Authors:
Andrey A. Poloznikov, Sergey V. Nikulin, Dmitry M. Hushpulian, Anna Yu. Khristichenko, Andrey I. Osipyants, Andrey F. Asachenko, Olga V. Shurupova, Svyatoslav S. Savin, Sue H. Lee, Irina N. Gaisina, Gregory R. J. Thatcher, Anthony Narciso, Eric P. Chang, Sergey V. Kazakov, Nancy Krucher, Vladimir I. Tishkov, Bobby Thomas, Irina G. GazaryanJournal:
Antioxidants
2021 Heading link
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Authors
Cutler T. Lewandowski, Md.Wasim Khan, Manel BenAissa, Oleksii Dubrovskyi, Martha Ackerman-Berrier, Mary Jo LaDu, Brian T. Layden, Gregory R.J. Thatcher
Journal
eBioMedicine
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Authors
Zhengnan Shen, Kiira Ratia, Laura Cooper, Deyu Kong, Hyun Lee, Youngjin Kwon, Yangfeng Li, Saad Alqarni, Fei Huang, Oleksii Dubrovskyi, Lijun Rong, Gregory R. J. Thatcher, and Rui Xiong
Journal
Journal of Medicinal Chemistry
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Authors
Oleksii Dubrovskyi, Erica Hasten, Steven M. Dudek, Michael T. Flavin, and Leo Li-Ying Chan
Journal
SLAS DISCOVERY: Advancing the Science of Drug Discovery
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Authors
Moushimi Amaya, Han Cheng, Viktoriya Borisevich, Chanakha K Navaratnarajah, Roberto Cattaneo, Laura Cooper, Terry W Moore, Irina N Gaisina, Thomas W Geisbert, Lijun Rong, and Christopher C Broder
Journal
Antiviral Research
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Authors
Ji-in Vivien Choi, Boriana K. Tchernookova, Wasan Kumar, Lech Kiedrowski, Calla Goeke, Marina Guizzetti, John Larson, Matthew A. Kreitzer and Robert Paul Malchow
Journal
Front. Cell. Neurosci
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Authors
Zhengnan Shen, Kiira Ratia, Laura Cooper, Deyu Kong, Hyun Lee, Youngjin Kwon, Yangfeng Li, Saad Alqarni, Fei Huang, Oleksii Dubrovskyi, Lijun Rong, Gregory Thatcher, Rui Xiong
Journal
ACS Pharmacolo. Transl. Sci.
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Authors
Sarah B. Scheinman, Steve Zaldua, Adedoyin Dada, Kateryna Krochmaliuk,
Katherine Dye, Felecia M. Marottoli, Gregory R. J. Thatcher and Leon M. TaiJournal
Frontiers in Neuroscience
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Authors
Adam Schager, Rui Xiong, Laura Cooper Raghad Nowar, Hyun Lee, Yangfeng Li,
Benjamin E. Ramirez, Norton P. Peet, Michael Caffrey, Gregory R.J. Thatcher, Erica Ollmann Saphire, Han Cheng, Lijun RongJournal
PLOS Pathogens
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Authors
Rachel C. Knopp Ammar Jastaniah, Oleksii Dubrovskyi, Irina Gaisina, Leon Tai
and Gregory R. J. ThatcherJournal
ACS Pharmacolo. Transl. Sci.
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Authors
Ruikun Du, Han Cheng, Qinghua Cui, Norton P Peet, Irina N Gaisina, and Lijun Rong
Journal
Antiviral Research
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Authors
Manel Ben Aissa, Cutler T. Lewandowski, Kiira M. Ratia, Sue J. Lee,
Brian T. Layden, Mary Jo LaDu and Gregory R. J. ThatcherJournal
ACS Pharmacolo. Transl. Sci.
2020 Heading link
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Authors
Aleksandar Antanasijevic, Matthew A Durst, Han Cheng, Irina N Gaisina, Jasmine T Perez, Balaji Manicassamy, Lijun Rong, Arnon Lavie, and Michael Caffrey
Journal
Life Science Alliance
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Authors
Yangfeng Li, Jiong Zhao, Lauren M. Gutgesell,
Zhengnan Shen, Kiira Ratia, Katherine Dye, Oleksii Dubrovskyi, Huiping Zhao, Fei Huang, Debra A. Tonetti, Gregory R. J. Thatcher, and Rui XiongJournal
J Med Chem
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Authors
Haining Lyu, Pavel A. Petukhov, Paul R. Banta
Ajit Jadhav, Wendy A. Lea, Qing Cheng, Elias S. J. Arnér, Anton Simeonov, Gregory R. J. Thatcher, Francesco Angelucci, David L. WilliamsJournal
Infectious Diseases
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Authors
Irina N. Gaisina, Norton P. Peet, Letitia Wong, Adam M. Schafer, Han Cheng, Manu Anantpadma, Robert A. Davey, Gregory R. J. Thatcher, and Lijun Rong
Journal
j Med Chem
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Authors
Cutler Lewandowski, Md. Wasim Khan, Manel Ben Aissa, Brian Layden
and Gregory ThatcherJournal
Circulation
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Authors
B. Abderrahman, PY Maximov, RF Curpan, JS Hanspal, P Fan, R Xiong, DA Tonetti,
GRJ Thatcher, VC JordanJournal
Molecular Pharmacology
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Authors
Rachel C. Knopp, Sue J. Lee, Michael Hollas, Emily Nepomuceno, David Gonzalez,
Kevin Tam, Daniyal Aamir, Yuiting Want, Emily Pierce, Manel Ben Aissa, Gregory R. J. TatcherJournal
ReDox Biology
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Authors
Ivan Pavlinov, Maryna Salkovski and Leslie N. Aldrich
Journal
J American Chemical Society
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Authors
Irina Gasina, Norton P. Peet, Han Cheng, Ping Li, Ruikun Du, Qinghua Cui,
Kevin Furlong, Balaji Manicassamy, Michael Caggrey, Gregory R. J. Thatcher, Lijun RongJournal
J Med Chem
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Authors
Ammar Jastaniah, Irina N Gaisina, Rachel C. Knopp, Gregory R. J. Thatcher
Journal
ChemMedChem
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Authors
Rachel C.Knopp, Sue H.Lee, Michael Hollas, Emily Nepomuceno, David Gonzalez, Kevin Tam,
Daniyal Aamir, Yueting Wang, Emily Pierce, Manel Ben Aissa, Gregory R.J. ThatcherJournal
Science Direct
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Authors
Laura Cooper, Adam Schafer, Yangfeng Li,
Han Cheng, Bani Medegan Fagla, Zhengnan Shen, Raghad Nowar, Katherine Dye, Manu Anantpadma, Robert A. Davey, Gregory RJ Thatcher, Lijun Rong, and Rui XiongJournal
J Med Chem
2019 Heading link
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Authors
Yunlong Lu, Lauren M. Gutgesell, Rui Xiong, Jiong Zhao, Yangfeng Li, Carlo I. Rosales, Michael Hollas, Zhengnan Shen, Jesse Gordon-Blake, Katherine Dye, Yueting Wang, Sue Lee, Hu Chen, Donghong He, Oleksii Dubrovyskyii, Huiping Zhao, Fei Huang, Amy W. Lasek, Debra A. Tonetti, and Gregory R. J. Thatcher
Journal
J Med Chem
2018 Heading link
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Authors
Manel Ben Aissa, Alycia F. Tipton, Zachariah Bertels, Ronak Gandhi,
Laura S. Moye, Madeline Novack, Brian M. Bennett, Yueting Wang, Vladislav Litosh, Sue H. Lee, Irina N. Gaisina, Gregory R. J. Thatcher Amynah A PradhanJournal
Cephalalgia
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Authors
Yao Yao, Chen Kong, Liang Yin, Atul D. Jain, Kiira Ratia, Gregory R. J. Thatcher,
Terry W. Moore, Tom G. Driver, Lawrence W. MillerJournal
Chemistry
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Authors
Tiara G Perez Morales, Kiira Ratia, Duo-Sheng Wang, Artemis Gogos,
Laura Bloem, Tom G. Driver, Michael J. FederleJournal
J. Biol Chem
2017 Heading link
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Authors
Rui Xiong, Jiong Zhao, Lauren M. Gutgesell, Yueting Wang, Sue Lee, Bhargava Karumudi, Huiping Zhao, Yunlong Lu, Debra A. Tonetti, and Gregory R. J. Thatcher
Journal
J Med Chem
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Authors
Abir Bhattacharjee, Antara Sinha, Kiira Ratia, Liang Yin, Loruhama Delgado-Rivera, Pavel A. Petukhov, Gregory R. J. Thatcher, Duncan J. Wardrop
Journal
ACS Med. Chem. Lett.
2016 Heading link
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Authors
Jia Luo, Sue H. Lee, Lawren VandeVrede, Zhihui Qin, Manel Ben Aissa, John Larson, Andrew F. Teich, Ottavio Arancio, Yohan D’Souza, Ahmed Elharram, Kevin Koster, Leon M. Tai, Mary Jo LaDu, Brian M. Bennett, and Gregory R. J. Thatcher
Journal
Molecular Neurodegeneration
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Authors
Rui Xiong, Hitisha K. Patel, Lauren M. Gutgesell, Jiong Zhao, Loruhama Delgado-Rivera, Thao N. D. Pham, Huiping Zhao, Kathryn Carlson, Teresa Martin, John A. Katzenellenbogen, Terry W. Moore, Debra A. Tonetti, and Gregory R. J. Thatcher
Journal
J Med Chem